Shun-Jun Ji*(纪顺俊)
Key Laboratory of Organic Synthesis of Jiangsu Province, College of Chemistry, Chemical Engineering and Materials Science, Soochow University, Suzhou 215123, China
J. Org. Chem. 2015, 80, 7928–7936
A palladium-catalyzed efficient C–H acylation reaction of biaryl-2-amines and aromatic aldehydes is developed. This dehydrogenative cross-coupling protocol could furnish monoacylation and diacylation products in moderate to good yields with a broad substrate scope and good regioselectivity.
链接:
//pubs.acs.org/doi/abs/10.1021/acs.joc.5b00962